SCHEMBL7302586

SCHEMBL7302586

COc1cccc2c1c(=O)[nH]c(=O)n2CCCCN1CC=C(c2ccccc2)CC1

nearest known ligand 0.75

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.75
HTR7 P34969 5/20 0.50
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CASP1 P29466 1/20 0.47
HBB P68871 1/20 0.47
USP2 O75604 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HTR1A P08908 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302722 0.87 PARP1 (0.79) PARP1
SCHEMBL7308205 0.87 PARP1 (0.64) PARP1HTR7KDM4EALDH1A1MAPT
SCHEMBL7300722 0.85 PARP1 (0.79) PARP1HTR7
SCHEMBL7309614 0.85 PARP1 (0.79) PARP1HTR7KDM4EMAPTHTR1A
SCHEMBL12231980 0.85 PARP1 (1.00) PARP1
SCHEMBL7307887 0.85 PARP1 (0.79) PARP1HTR7HTR1A
Hydrochloric Acid SCHEMBL7301292 0.85 PARP1 (0.98) PARP1
SCHEMBL7299268 0.82 PARP1 (0.73) PARP1
SCHEMBL7305161 0.82 PARP1 (0.73) PARP1
SCHEMBL7308137 0.80 PARP1 (0.60) PARP1KDM4EALDH1A1CASP1HBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed