SCHEMBL7308205

SCHEMBL7308205

COc1cc2c(=O)[nH]c(=O)n(CCCCN3CC=C(c4ccccc4)CC3)c2cc1OC

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.64
CASP1 P29466 1/20 0.58
HBB P68871 1/20 0.58
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 2/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
USP2 O75604 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 1/20 0.54
HTR7 P34969 1/20 0.48
HTR1A P08908 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303980 0.88 PARP1 (0.60) PARP1CASP1HBBKDM4EALDH1A1
SCHEMBL7308137 0.88 PARP1 (0.60) PARP1CASP1HBBKDM4EALDH1A1
SCHEMBL7302586 0.87 PARP1 (0.75) PARP1CASP1HBBKDM4EALDH1A1
SCHEMBL7303316 0.85 PARP1 (0.64) PARP1MAPTTDP1TSHRHTR1A
Bromide SCHEMBL7303725 0.85 PARP1 (0.63) PARP1MAPTTDP1TSHRHTR1A
SCHEMBL7305161 0.84 PARP1 (0.73) PARP1
SCHEMBL7307656 0.83 PARP1 (0.63) PARP1MAPTTDP1TSHRHTR1A
SCHEMBL7302855 0.83 PARP1 (0.64) PARP1
SCHEMBL7308221 0.83 PARP1 (0.63) PARP1
Hydrochloric Acid SCHEMBL7301544 0.83 PARP1 (0.63) PARP1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed