SCHEMBL7302955

SCHEMBL7302955

COC(=O)COc1ccc(C(O)CNC(=O)c2ccc(C(=N)N)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
ITGB3 P05106 3/20 0.46
ITGA2B P08514 3/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAPT P10636 1/20 0.43
POLB P06746 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PRSS1 P07477 2/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
F10 P00742 1/20 0.41
ADRB3 P13945 2/20 0.41
GLA P06280 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9266142 0.99 ALDH1A1 (0.46) ALDH1A1ITGB3ITGA2BNPC1RAB9A
SCHEMBL7298011 0.88 ITGB3 (0.57) ALDH1A1ITGB3ITGA2BNPC1RAB9A
Hydrochloric Acid SCHEMBL9270840 0.87 ITGB3 (0.45) ALDH1A1ITGB3ITGA2BHPGDNPSR1
Hydrochloric Acid SCHEMBL9270834 0.87 ITGB3 (0.45) ALDH1A1ITGB3ITGA2BHPGDNPSR1
SCHEMBL9269322 0.84 MEN1 (0.51) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL9271047 0.84 MEN1 (0.51) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Hydrochloric Acid SCHEMBL9270105 0.84 HPGD (0.43) ALDH1A1ITGB3ITGA2BHPGDNPSR1
Hydrochloric Acid SCHEMBL9270097 0.84 HPGD (0.43) ALDH1A1ITGB3ITGA2BHPGDNPSR1
SCHEMBL7301011 0.83 POLB (0.57) ALDH1A1SMN1; SMN2POLBADRB3GLA
Hydrochloric Acid SCHEMBL9265744 0.82 POLB (0.56) ALDH1A1SMN1; SMN2POLBADRB3GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US claimed