SCHEMBL7303025

SCHEMBL7303025

N#CC(CCCN1CCC(C(=O)c2ccc(F)cc2)CC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.63
KDM4E B2RXH2 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63
CCR1 P32246 1/20 0.61
CCR3 P51677 1/20 0.58
HTR2C P28335 1/20 0.55
HTR7 P34969 1/20 0.55
HTR6 P50406 1/20 0.55
KCNA3 P22001 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9374606 0.99 HTR2A (0.62) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9586092 0.89 CYP2D6 (0.51) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9374406 0.85 HTR2A (0.58) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9374768 0.84 HTR2A (0.57) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9585725 0.83 KCNH2 (0.60) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9585669 0.81 HTR2A (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9103936 0.79 KCNA3 (0.85) CCR1CCR3KCNA3
SCHEMBL9374226 0.79 HTR2A (0.51) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9672004 0.78 HTR2A (0.66) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9374947 0.78 HSD11B1 (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294183-B1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO KK (JP) 1994-03-30 EP claimed
EP-0294183-A1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO CO., INC. (JP) 1988-12-07 EP claimed
US-5229400-A Cardiovascular disorders AJINOMOTO CO., INC. (JP) 1993-07-20 US disclosed
EP-0479601-A2 Piperidine derivatives and their use as antiarrhythmic agents Ajinomoto Co., Inc. (JP) 1992-04-08 EP disclosed
EP-0294183-A1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO CO., INC. (JP) 1988-12-07 EP disclosed