SCHEMBL7303933

SCHEMBL7303933

CC(C)(C)ONC(=O)C(CS(=O)(=O)c1ccc(Oc2ccccc2)cc1)NC(=O)OCc1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 13/20 0.76
CTSK P43235 4/20 0.48
CTSS P25774 2/20 0.48
MMP1 P03956 1/20 0.46
MMP2 P08253 1/20 0.46
CA1 P00915 1/20 0.46
CA5A P35218 1/20 0.46
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303925 1.00 MMP13 (0.76) MMP13CTSKCTSSMMP1MMP2
SCHEMBL7310335 0.92 MMP13 (0.65) MMP13CTSKCTSSMMP1MMP2
SCHEMBL7308069 0.87 MMP13 (1.00) MMP13CTSKCTSSMMP1
SCHEMBL7308056 0.87 MMP13 (1.00) MMP13CTSKCTSSMMP1
SCHEMBL7180333 0.85 MMP13 (0.82) MMP13CTSKCTSSMMP1
SCHEMBL7308292 0.82 MMP13 (0.61) MMP13MMP1MMP2
SCHEMBL7302646 0.81 CA2 (0.52) MMP13CTSKCTSSCTSLCTSB
SCHEMBL7302654 0.81 CA2 (0.52) MMP13CTSKCTSSCTSLCTSB
SCHEMBL7299964 0.80 MMP13 (0.82) MMP13CTSKCTSSMMP1MMP2
SCHEMBL7301636 0.79 MMP13 (0.57) MMP13MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed