SCHEMBL7304372

SCHEMBL7304372

O=CN(OCc1ccccc1)c1ccc(O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.44
LMNA P02545 2/20 0.44
CYP2C19 P33261 2/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
PTGS2 P35354 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HIF1A Q16665 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
CA12 O43570 1/20 0.42
AKR1B10 O60218 1/20 0.42
AKR1B1 P15121 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
FNTA P49354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936315 0.90 TSHR (0.41) CYP1A2CYP2C19SLC6A2SLC6A3CA9
SCHEMBL9005245 0.85 MAOA (0.43) LMNACA12AKR1B10AKR1B1CA4
SCHEMBL10750641 0.85 TSHR (0.35) CYP1A2CYP2C19SLC6A2SLC6A3CA9
SCHEMBL27478897 0.84 TSHR (0.34) SLC6A2SLC6A3CA9ALDH1A1MAPT
SCHEMBL11185353 0.83 ALDH1A1 (0.43) LMNASLC6A2SLC6A3ABCG2ALDH1A1
SCHEMBL5614230 0.82 TSHR (0.36) CYP2C19SLC6A2SLC6A3CA9ALDH1A1
SCHEMBL2409895 0.78 ALDH1A1 (0.48) CYP1A2LMNACYP2C19SLC6A2SLC6A3
SCHEMBL28253562 0.77 ESR1 (0.39) LMNASLC6A2HDAC6CA12CA7
SCHEMBL28253465 0.77 ESR1 (0.39) LMNASLC6A2HDAC6CA12CA7
SCHEMBL9626473 0.77 MEN1 (0.36) LMNAALDH1A1MAPTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed