SCHEMBL7304645

SCHEMBL7304645

CC(C)(C)OC(=O)N1CCCC(C(=O)NCCC(=O)OCc2ccccc2)C1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.60
ITGA2B P08514 4/20 0.60
HTT P42858 1/20 0.52
RAB9A P51151 2/20 0.52
ALDH1A1 P00352 2/20 0.52
NPC1 O15118 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
HPGD P15428 1/20 0.52
KMT2A Q03164 2/20 0.48
GAA P10253 1/20 0.48
STS P08842 1/20 0.47
USP30 Q70CQ3 2/20 0.47
MEN1 O00255 1/20 0.46
F2R P25116 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303090 0.94 HTT (0.59) ITGB3ITGA2BHTTRAB9ANPC1
SCHEMBL7500520 0.92 ITGB3 (0.55) ITGB3ITGA2BHTTRAB9AALDH1A1
SCHEMBL22616973 0.86 ALDH1A1 (0.69) HTTRAB9AALDH1A1NPC1CYP3A4
SCHEMBL2433449 0.85 USP30 (0.54) ITGB3ITGA2BHTTKMT2ASTS
SCHEMBL2433452 0.85 USP30 (0.54) ITGB3ITGA2BHTTKMT2ASTS
SCHEMBL7290589 0.84 CHRM1 (0.51) ITGB3ITGA2BALDH1A1HPGDKMT2A
SCHEMBL22616979 0.84 GAA (0.67) RAB9AALDH1A1NPC1CYP3A4CYP2D6
SCHEMBL22617001 0.84 GAA (0.67) RAB9AALDH1A1NPC1CYP3A4CYP2D6
SCHEMBL2263064 0.83 ITGB3 (0.58) ITGB3ITGA2BHTTRAB9ANPC1
SCHEMBL2263069 0.83 ITGB3 (0.58) ITGB3ITGA2BHTTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed