SCHEMBL7304804

SCHEMBL7304804

CC(C)(C)OC(=O)NCCNC(=O)Cc1ccc(C2=NNC(=O)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 6/20 0.47
PDE3A Q14432 5/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
MIF P14174 1/20 0.43
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KCNH2 Q12809 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
BCHE P06276 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
PDE2A O00408 1/20 0.36
PDE1A P54750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297671 0.81 PDE3B (0.53) PDE3BPDE3AMAPTLMNANPY1R
SCHEMBL18522739 0.75 MAPT (0.41) PDE3BPDE3AMAPTLMNANPY1R
SCHEMBL15284610 0.74 ESRRB (0.58) MAPTLMNAMIFSMN1; SMN2CA1
SCHEMBL14679418 0.74 HPGD (0.57) MAPTLMNAKMT2ACA1CA2
SCHEMBL14155336 0.73 LMNA (0.56) LMNAKMT2ASMN1; SMN2CA1CA2
SCHEMBL4881326 0.72 PDE3B (0.42) PDE3BPDE3ALMNASMN1; SMN2PDE4A
SCHEMBL8339349 0.72 SMN1; SMN2 (0.55) PDE3BPDE3AMAPTLMNANPY1R
SCHEMBL14679377 0.70 HPGD (0.62) MAPTLMNAKMT2ACA1CA2
SCHEMBL10474306 0.70 MAPT (0.65) PDE3BPDE3AMAPTLMNANPY1R
SCHEMBL7240480 0.69 BCL2 (0.53) MAPTLMNAKMT2ABCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed