SCHEMBL7305489

SCHEMBL7305489

Cc1cccc(NC(=O)c2ccccc2)c1Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.72
POLB P06746 2/20 0.72
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
MAPT P10636 3/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
LMNA P02545 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
HDAC1 Q13547 2/20 0.57
HDAC3 O15379 1/20 0.57
MAPK1 P28482 1/20 0.57
HDAC2 Q92769 1/20 0.57
CYP1A2 P05177 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
MDM4 O15151 1/20 0.53
TP53 P04637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790102 0.88 NPC1 (0.68) HPGDPOLBNPC1RAB9AMAPT
N-O-Tolylbenzamide SCHEMBL3223289 0.84 HPGD (1.00) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL4094232 0.83 HDAC1 (0.72) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL7264464 0.83 POLB (0.77) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL11769542 0.83 POLB (0.77) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL9621459 0.83 MEN1 (0.82) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL30288146 0.83 POLB (0.77) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL13602430 0.81 MAPT (0.56) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL14492571 0.81 KCNK3 (0.63) HPGDPOLBNPC1RAB9AMAPT
SCHEMBL16330055 0.80 POLB (0.72) HPGDPOLBNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022089406-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海青煜医药科技有限公司 2022-05-05 WO disclosed
US-5412099-A Intermediate benzothiazolyl- and benzoxazolyl-aldehyde compounds BAYER AKTIENGESELLSCHAFT (DE) 1995-05-02 US disclosed
EP-0450420-B1 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1994-09-21 EP disclosed
US-5254692-A Inotropic BAYER AKTIENGESELLSCHAFT (DE) 1993-10-19 US disclosed
US-5200420-A Inotropic agents for cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
EP-0450420-A2 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1991-10-09 EP disclosed