Iodide

Iodide

SCHEMBL7305544

C=CC[N+]1(C)CCN(c2nc3ccc(OC)cc3o2)CC1.[I-]

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.36
GABRP O00591 4/20 0.44
GABRD O14764 4/20 0.44
GABRA1 P14867 4/20 0.44
GABRB1 P18505 4/20 0.44
GABRG2 P18507 4/20 0.44
GABRB3 P28472 4/20 0.44
GABRA5 P31644 4/20 0.44
GABRA3 P34903 4/20 0.44
GABRA2 P47869 4/20 0.44
GABRB2 P47870 4/20 0.44
GABRA4 P48169 4/20 0.44
GABRE P78334 4/20 0.44
GABRA6 Q16445 4/20 0.44
GABRG1 Q8N1C3 4/20 0.44
GABRG3 Q99928 4/20 0.44
GABRQ Q9UN88 4/20 0.44
F2RL3 Q96RI0 2/20 0.37
APP P05067 1/20 0.37
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL7306788 0.85 ESR1 (0.36) APPGAAKMT2A
Bromide SCHEMBL6488179 0.84 KDM4E (0.41) GABRPGABRDGABRA1GABRB1GABRG2
Iodide SCHEMBL7307948 0.84 PRKDC (0.38) FAAHGAAKMT2A
Iodide SCHEMBL7307306 0.82 SORD (0.47) HCRTR1HCRTR2TSHRGAAKMT2A
Iodide SCHEMBL7305936 0.81 NPC1 (0.40) ALDH1A1L3MBTL1GAAKMT2A
Hydrochloric Acid SCHEMBL7305474 0.80 SORD (0.47) TSHRGAAKMT2A
SCHEMBL7340538 0.79 NPC1 (0.41) ALDH1A1L3MBTL1GAAKMT2A
Iodide SCHEMBL7304275 0.78 SORD (0.44) HCRTR1HCRTR2TSHRGAAKMT2A
Iodide SCHEMBL6501966 0.78 PTGES (0.46)
Bromide SCHEMBL6488073 0.78 PIK3CB (0.38) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0621271-B1 Benzoxazole derivatives and their use as serotonin 5-HT3 receptor antagonists MEIJI SEIKA KAISHA (JP) 2001-10-17 EP disclosed
US-5631257-A ANTISEROTONIN AGENTS FOR TREATMENT OF NAUSEA AND ANTIEMETICS MEIJI SEIKA KAISHA, LTD. (JP) 1997-05-20 US disclosed
EP-0621271-A1 Benzoxazole derivatives and their use as serotonin 5-HT3 receptor antagonists MEIJI SEIKA KAISHA LTD. (JP) 1994-10-26 EP disclosed