SCHEMBL7305959

SCHEMBL7305959

CCCCc1nc(C(=O)OCc2ccc(-c3ccccc3-c3nnnn3C(c3ccccc3)(c3ccccc3)c3ccccc3)cc2)c(C(C)O)n1CC

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGT P01019 2/20 0.52
AGTR1 P30556 5/20 0.48
AGTR2 P50052 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306141 0.96 AGTR1 (0.52) AGTAGTR1AGTR2
SCHEMBL7310916 0.88 AGT (0.51) AGTAGTR1AGTR2
SCHEMBL7306983 0.87 AGTR1 (0.49) AGTAGTR1AGTR2
SCHEMBL7299142 0.87 AGT (0.50) AGTAGTR1AGTR2
SCHEMBL7303265 0.84 AGTR1 (0.54) AGTAGTR1AGTR2
SCHEMBL1988059 0.84 AGTR1 (0.54) AGTAGTR1AGTR2
SCHEMBL7299320 0.84 AGT (0.49) AGTAGTR1AGTR2
SCHEMBL7312738 0.83 AGTR2 (0.53) AGTAGTR1AGTR2
SCHEMBL9385090 0.81 AGT (0.61) AGTAGTR1AGTR2
SCHEMBL7307299 0.81 AGTR1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545912-B1 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0545912-A2 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1993-06-09 EP disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed