SCHEMBL7306066

SCHEMBL7306066

Cn1nc(-c2cccc(C(F)(F)F)c2)n(C)c1=S

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GABRA1 P14867 1/20 0.45
HPGD P15428 1/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA5 P31644 1/20 0.45
GABRA3 P34903 1/20 0.45
GABRA2 P47869 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
KCNH2 Q12809 1/20 0.44
PTGS2 P35354 1/20 0.43
POLB P06746 1/20 0.42
IKBKB O14920 1/20 0.42
BRD4 O60885 1/20 0.42
PIN1 Q13526 1/20 0.41
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14077013 0.74 KDM4E (0.55) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL6915245 0.73 KDM4E (0.48) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL7435538 0.72 GRM5 (0.38) HSD17B10ALDH1A1CYP1A2CYP3A4KCNH2
SCHEMBL1720026 0.71 PTGS2 (0.49) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL1720476 0.71 PTGS2 (0.49) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL27888810 0.70 PTGS2 (0.46) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL27888812 0.70 KMT2A (0.51) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL2662898 0.70 PTPN5 (0.62) KDM4EHSD17B10ALDH1A1IKBKBBRD4
SCHEMBL12832618 0.70 NPC1 (0.47) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL22633138 0.70 TLR8 (0.51) KDM4EHSD17B10ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452926-B1 5-aryl-4-alkyl-3H-1,2,4-triazole-3-thiones useful as memory enhancers MERRELL DOW PHARMA (US) 1996-03-13 EP disclosed