SCHEMBL7435538

SCHEMBL7435538

Cn1nc(-c2ccc(F)c(F)c2)n(C)c1=S

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.38
PTGS2 P35354 2/20 0.36
OPRL1 P41146 1/20 0.35
ALDH1A1 P00352 2/20 0.35
APOBEC3G Q9HC16 1/20 0.35
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DRD3 P35462 2/20 0.34
KCNH2 Q12809 2/20 0.34
NOTUM Q6P988 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
TYMP P19971 1/20 0.33
TGFBR1 P36897 1/20 0.33
PGR P06401 1/20 0.33
PTGS1 P23219 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299383 0.81 ALDH1A1 (0.43) GRM5ALDH1A1APOBEC3GHSD17B10MAPT
Suritozole SCHEMBL121081 0.79 RXFP1 (0.43) PTGS2ALDH1A1APOBEC3GCYP1A2HSD17B10
SCHEMBL7306147 0.77 MAPT (0.50) GRM5ALDH1A1APOBEC3GUSP2NOTUM
SCHEMBL7485829 0.77 LMNA (0.50) GRM5ALDH1A1APOBEC3GCYP1A2CYP3A4
SCHEMBL7304540 0.73 KDM4E (0.40) GRM5CYP3A4PGR
SCHEMBL7297002 0.72 TDP1 (0.45) ALDH1A1APOBEC3GHSD17B10
SCHEMBL7302275 0.72 ALDH1A1 (0.33) ALDH1A1RAB9AMAPTCYP11B1CYP11B2
SCHEMBL2311265 0.72 ALDH1A1 (0.66) ALDH1A1APOBEC3GHSD17B10MAPT
SCHEMBL7306066 0.72 KDM4E (0.45) PTGS2ALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9833680 0.72 MEN1 (0.42) GRM5ALDH1A1HSD17B10MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4775688-A 5-aryl-2,4-dialkyl-3H-1,2,4-triazole-3-thiones and their use as antidepressants MERRELL DOW PHARMACEUTICALS INC. (US) 1988-10-04 US claimed
US-4775688-A 5-aryl-2,4-dialkyl-3H-1,2,4-triazole-3-thiones and their use as antidepressants MERRELL DOW PHARMACEUTICALS INC. (US) 1988-10-04 US disclosed
EP-0221485-A1 5-Aryl-2,4-dialkyl-3H-1,2,4-triazole-3-thiones and their use as antidepressants MERRELL DOW PHARMACEUTICALS INC. (US) 1987-05-13 EP disclosed