SCHEMBL7306289

SCHEMBL7306289

O=C(O)C(=O)[C@@H]1CCCN1C(=O)CCC(=O)N(Cc1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 12/20 0.47
ALDH1A1 P00352 3/20 0.45
NPC1 O15118 1/20 0.45
GLA P06280 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
PAX8 Q06710 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ACE2 Q9BYF1 1/20 0.44
CPT2 P23786 1/20 0.43
CPT1A P50416 1/20 0.43
CHRM2 P08172 2/20 0.42
CHRM1 P11229 2/20 0.42
CHRM3 P20309 2/20 0.42
F2 P00734 1/20 0.41
MEN1 O00255 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283951 0.93 F2 (0.43) ACEALDH1A1NPC1GLAHTT
SCHEMBL9484859 0.92 ACE (0.56) ACEACE2CHRM2CHRM1CHRM3
SCHEMBL7281408 0.90 DPP4 (0.43) ACEACE2
SCHEMBL9178463 0.89 ACE (0.43) ACEALDH1A1SMN1; SMN2ACE2CPT2
SCHEMBL7282427 0.85 NPC1 (0.56) ACENPC1HTTRAB9ASMN1; SMN2
SCHEMBL7267053 0.84 ALDH1A1 (0.45) ACEALDH1A1NPC1GLAHTT
Water SCHEMBL7282829 0.84 NPC1 (0.55) ACENPC1HTTRAB9ASMN1; SMN2
SCHEMBL7283585 0.82 MEN1 (0.52) ACENPC1HTTRAB9AACE2
SCHEMBL7290889 0.81 CHRM2 (0.43) ACEALDH1A1NPC1GLAHTT
SCHEMBL8994520 0.81 KDM4E (0.44) ACEALDH1A1SMN1; SMN2ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537802-B1 N-acylpyrrolidines, process for their preparation and their use for prevention and/or treatment of amnesia ONO PHARMACEUTICAL CO (JP) 1999-08-25 EP claimed
US-5545657-A 1-ALKYLOYLPYRROLIDIN-2-YLOXOALKANOIC ACIDS AND DERIVATIVES; ANTIAMNESIA AGENTS; INHIBITORS OF PROLYL ENDOPEPTIDASE; SUPPRESSION OF NEUROTRANSMITTER METABOLISM ONO PHARMACEUTICAL CO., LTD. (JP) 1996-08-13 US claimed
EP-0537802-A2 N-acylpyrrolidines and N-acylthiazolidines, process for their preparation and their use for prevention and/or treatment of amnesia ONO PHARMACEUTICAL CO., LTD. (JP) 1993-04-21 EP claimed
EP-0345428-A1 Anti-amnesic pyrrolidine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1989-12-13 EP claimed