SCHEMBL7306807

SCHEMBL7306807

O=C(N[C@@H](Cc1ccccc1)[C@H](O)CN1CC[C@@H]2CCCC[C@@H]2[C@@H]1C(F)(F)F)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
CTSB P07858 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
OPRK1 P41145 2/20 0.40
ACE P12821 1/20 0.40
KLK5 Q9Y337 1/20 0.40
CASP1 P29466 3/20 0.39
HRH1 P35367 1/20 0.39
CTRB1 P17538 2/20 0.38
KDM1A O60341 4/20 0.38
PREP P48147 2/20 0.38
MAOA P21397 2/20 0.38
RCOR1 Q9UKL0 2/20 0.38
KDM1B Q8NB78 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304137 1.00 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1CTSB
SCHEMBL7307601 0.90 ADORA3 (0.64) ADORA3ADORA2AADORA2BADORA1OPRK1
SCHEMBL7305767 0.90 ADORA3 (0.64) ADORA3ADORA2AADORA2BADORA1OPRK1
SCHEMBL9168915 0.83 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1OPRK1
SCHEMBL9168426 0.83 ADORA3 (0.46) ADORA3ADORA2AADORA2BADORA1OPRK1
SCHEMBL7312690 0.80 MEN1 (0.37)
SCHEMBL7300465 0.78 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1CTSB
SCHEMBL9018608 0.78 ADORA3 (0.45) ADORA3ADORA2AADORA2BADORA1CTSB
SCHEMBL7389742 0.78 ADORA3 (0.55) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL7267808 0.76 ADORA3 (0.62) ADORA3ADORA2AADORA2BADORA1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed