SCHEMBL7300465

SCHEMBL7300465

O=C(N[C@@H](Cc1ccccc1)[C@H](O)CN1CCC(=O)C1C(F)(F)F)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
CASP1 P29466 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.44
CTSB P07858 9/20 0.44
CTSK P43235 6/20 0.42
CTSS P25774 5/20 0.42
CTRB1 P17538 2/20 0.42
CTSL P07711 4/20 0.41
ELANE P08246 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304097 0.79 ADORA3 (0.47) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL7309658 0.79 ADORA3 (0.47) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL7306807 0.78 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL7304137 0.78 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL5704587 0.75 TRPM8 (0.57) TRPM8CTSBCTSKCTSSCTRB1
SCHEMBL9018608 0.75 ADORA3 (0.45) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL7268961 0.74 TRPM8 (0.54) TRPM8CTSBCTSKCTSSCTRB1
SCHEMBL7267808 0.74 ADORA3 (0.62) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL7302736 0.73 ADORA3 (0.73) ADORA3ADORA2AADORA2BADORA1CASP1
SCHEMBL7428630 0.73 TRPM8 (0.55) TRPM8CTSBCTSKCTSSCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed