SCHEMBL7306893

SCHEMBL7306893

O=C(O)CCN1CCN(CC2CN(C3CCNCC3)C(=O)O2)CC1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 6/20 0.49
GLA P06280 1/20 0.35
CACNA2D1 P54289 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNB1 Q02641 1/20 0.34
ITGB3 P05106 5/20 0.34
ITGA2B P08514 5/20 0.34
KDM1A O60341 1/20 0.30
SMYD3 Q9H7B4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313924 0.88 HTR2B (0.51) HTR2BCACNA2D1CACNA1BCACNB1ITGB3
SCHEMBL7305444 0.87 HTR2B (0.50) HTR2BGLACACNA2D1CACNA1BCACNB1
SCHEMBL7304864 0.87 HTR2B (0.43) HTR2BITGB3ITGA2B
SCHEMBL7310988 0.83 HTR2B (0.52) HTR2BGLA
SCHEMBL7308191 0.82 HTR2B (0.46) HTR2BGLAITGB3ITGA2B
SCHEMBL7310427 0.81 HTR2B (0.43) HTR2B
SCHEMBL7305773 0.81 HTR2B (0.54) HTR2B
SCHEMBL7303482 0.81 HTR2B (0.48) HTR2BCACNA2D1CACNA1BCACNB1KDM1A
SCHEMBL7313313 0.80 HTR2B (0.45) HTR2BCACNA2D1CACNA1BCACNB1ITGB3
SCHEMBL7314426 0.77 HTR2B (0.50) HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP claimed
JP-8208629-A None JP disclosed
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
JP-H08208629-A ADHESION RECEPTOR ANTAGONISTIC COMPOUND MERCK PATENT GMBH 1996-08-13 JP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed