SCHEMBL7305773

SCHEMBL7305773

O=C(O)CCN1CCN(CC2CN(C3CCN(Cc4ccccc4)CC3)C(=O)O2)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.54
CHRM2 P08172 4/20 0.46
CHRM3 P20309 4/20 0.46
SIGMAR1 Q99720 4/20 0.44
ABCB1 P08183 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
KMT2A Q03164 1/20 0.44
HTR1A P08908 3/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
HTR7 P34969 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
FAAH O00519 1/20 0.43
CCR8 P51685 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306400 0.94 HTR2B (0.53) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7305604 0.90 HTR2B (0.56) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7307163 0.89 HTR2B (0.50) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7304924 0.89 HTR2B (0.49) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7306441 0.86 HTR2B (0.48) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7316544 0.85 ACHE (0.44) HTR2BSIGMAR1ABCB1KMT2AHTR1A
SCHEMBL7317110 0.84 SIGMAR1 (0.47) HTR2BSIGMAR1ABCB1KMT2AHTR1A
SCHEMBL7305444 0.84 HTR2B (0.50) HTR2BSIGMAR1
SCHEMBL7303558 0.83 HTR2B (0.52) HTR2BCHRM2CHRM3SIGMAR1ABCB1
SCHEMBL7308439 0.83 ACHE (0.50) FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed