SCHEMBL7306933

SCHEMBL7306933

COc1ccc(SC(N)=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.55
CA2 P00918 5/20 0.55
PARP10 Q53GL7 2/20 0.55
PARP1 P09874 1/20 0.55
PARP2 Q9UGN5 1/20 0.55
PARP4 Q9UKK3 1/20 0.55
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
HPGD P15428 1/20 0.51
PTGIR P43119 1/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP1B1 Q16678 1/20 0.46
F3 P13726 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229538 0.81 MAPT (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL9478248 0.79 PTGIR (0.59) CA1CA2PARP10PARP1PARP2
SCHEMBL11568437 0.79 HPGD (0.51) CA1CA2PARP10PARP1PARP2
SCHEMBL11711919 0.78 PARP10 (0.38) PARP10PARP4ALDH1A1MAPTHPGD
SCHEMBL20749917 0.78 PTGIR (0.49) CA1CA2PARP10PARP1PARP2
SCHEMBL28338045 0.78 CA1 (0.50) CA1CA2PARP10PARP1PARP2
SCHEMBL11569353 0.77 HPGD (0.46) CA1CA2PARP10PARP1PARP2
SCHEMBL11338721 0.76 ALDH1A1 (0.49) CA1CA2PARP10PARP1PARP2
SCHEMBL11768736 0.76 PLK1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL22735096 0.76 ALDH1A1 (0.49) CA1CA2PARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5674864-A ANALGESICS; ENDOPEPTIDASE AND ENKEPHALINASE INHIBITORS; CARDIOTONIC, PSYCHOTROPIC AND HYPERTENSIVE AGENTS ROUSSEL UCLAF (FR) 1997-10-07 US disclosed
EP-0742201-A1 PROCESS FOR PRODUCING AROMATIC OR HETEROAROMATIC SULFUR COMPOUNDS SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 1996-11-13 EP disclosed
EP-0465369-B1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1994-04-13 EP disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed
EP-0465369-A1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1992-01-08 EP disclosed