SCHEMBL7306947

SCHEMBL7306947

COc1ccc(NC(O)=S)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.69
CYP2C19 P33261 2/20 0.69
HPGD P15428 2/20 0.66
NPC1 O15118 7/20 0.65
RAB9A P51151 7/20 0.65
SMN1; SMN2 Q16637 5/20 0.65
MAPT P10636 6/20 0.62
ALDH1A1 P00352 6/20 0.62
MEN1 O00255 1/20 0.62
HTT P42858 1/20 0.62
KMT2A Q03164 1/20 0.62
MAOB P27338 3/20 0.61
MAOA P21397 2/20 0.61
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
GAA P10253 3/20 0.58
TDP1 Q9NUW8 3/20 0.56
LMNA P02545 2/20 0.56
TP53 P04637 1/20 0.55
ALOX15 P16050 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluoride SCHEMBL28392203 0.98 CYP1A2 (0.67) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL8167087 0.84 CYP1A2 (0.85) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL13715007 0.83 HPGD (0.66) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL1259295 0.82 CYP1A2 (1.00) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL4499854 0.81 HPGD (0.63) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL526026 0.81 ALDH1A1 (0.70) CYP1A2CYP2C19HPGDNPC1RAB9A
Hydrogen Sulfide SCHEMBL28246712 0.80 CYP1A2 (0.96) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL8977748 0.80 CYP1A2 (0.61) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL8531717 0.79 MAPT (0.64) CYP1A2CYP2C19HPGDNPC1RAB9A
SCHEMBL10624822 0.79 NPC1 (0.86) CYP1A2CYP2C19HPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9550790-B2 Thienopyranones as kinase inhibitors SIGNALRX PHARMACEUTICALS, INC. (US) 2017-01-24 US disclosed
US-5674864-A ANALGESICS; ENDOPEPTIDASE AND ENKEPHALINASE INHIBITORS; CARDIOTONIC, PSYCHOTROPIC AND HYPERTENSIVE AGENTS ROUSSEL UCLAF (FR) 1997-10-07 US disclosed
US-5637731-A CHOLINERGIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-06-10 US disclosed
US-5550257-A TREATING CENTRAL CHOLINERGIC DYSFUNCTION AMERICAN CYANAMID COMPANY (US) 1996-08-27 US disclosed
EP-0465369-B1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1994-04-13 EP disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed
EP-0465369-A1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1992-01-08 EP disclosed