SCHEMBL7307433

SCHEMBL7307433

O=c1[nH]c(=O)n(CCCCN2CC=C(c3ccc(Cl)cc3)CC2)c2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.62
SIGMAR1 Q99720 1/20 0.58
HTR1A P08908 1/20 0.52
HTR7 P34969 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305161 0.92 PARP1 (0.73) PARP1
SCHEMBL7299748 0.91 PARP1 (0.63) PARP1
SCHEMBL7308221 0.88 PARP1 (0.63) PARP1SIGMAR1
SCHEMBL7302855 0.88 PARP1 (0.64) PARP1SIGMAR1
SCHEMBL7299419 0.84 SIGMAR1 (0.58) PARP1SIGMAR1HTR1AHTR7
SCHEMBL7298835 0.84 KDM4E (0.53) PARP1SIGMAR1
SCHEMBL6621419 0.82 PARP1 (0.56) PARP1SIGMAR1HTR1AHTR7
SCHEMBL7300294 0.81 PARP1 (0.62) PARP1
SCHEMBL7307887 0.81 PARP1 (0.79) PARP1SIGMAR1HTR1AHTR7
Hydrochloric Acid SCHEMBL7301544 0.80 PARP1 (0.63) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed