SCHEMBL7307485

SCHEMBL7307485

Cc1nc(-c2ccc(N3CC(CO)OC3=O)cc2)no1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.52
MAOB P27338 2/20 0.52
CALML3 P27482 6/20 0.48
THRB P10828 1/20 0.45
DGAT1 O75907 1/20 0.43
GRM2 Q14416 3/20 0.43
P2RX3 P56373 2/20 0.43
MAPK14 Q16539 1/20 0.43
PLK1 P53350 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7385835 0.88 F10 (0.50) THRBDGAT1GRM2P2RX3
SCHEMBL7068870 0.88 THRB (0.47) MAOAMAOBTHRBDGAT1GRM2
SCHEMBL7387512 0.86 PLK1 (0.43) MAOATHRBDGAT1GRM2P2RX3
SCHEMBL27442648 0.84 S1PR1 (0.49) MAOAMAOBCALML3DGAT1GRM2
SCHEMBL7388767 0.84 SIGMAR1 (0.45) THRBDGAT1
SCHEMBL7309052 0.83 THRB (0.43) THRBGRM2P2RX3
SCHEMBL7387106 0.83 CA12 (0.44) THRBDGAT1GRM2P2RX3
SCHEMBL14183599 0.83 CALML3 (0.64) MAOAMAOBCALML3
SCHEMBL5530617 0.82 SIGMAR1 (0.45) THRBDGAT1
SCHEMBL7457616 0.81 PLK1 (0.45) THRBDGAT1P2RX3MAPK14PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5627197-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-05-06 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed