SCHEMBL7307825

SCHEMBL7307825

C=C1C[C@@H]2C(=O)NC(=O)[C@@H]2C1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.33
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2984006 1.00 MAP3K14 (0.33) MAP3K14CRBN
SCHEMBL10400960 0.72 CRBN (0.36) MAP3K14CRBN
SCHEMBL5909391 0.71 MAP3K14 (0.55) MAP3K14CRBN
SCHEMBL18545242 0.69 MAP3K14 (0.33) MAP3K14CRBN
SCHEMBL455753 0.69
SCHEMBL3628793 0.69 MAP3K14 (0.33) MAP3K14CRBN
SCHEMBL14139685 0.69
SCHEMBL25366289 0.69 POLB (0.35) MAP3K14CRBN
SCHEMBL17432744 0.67 BRD4 (0.41) MAP3K14CRBN
SCHEMBL7298906 0.67 KDM4E (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454121-B1 Azatetracyclic compounds SEARLE & CO (US) 1996-11-13 EP disclosed
US-5223613-A Prepared from cyclopenta(c)pyrrole derivatives; drug intermediates; antiemetics, anixiolytics G. D. SEARLE & CO. (US) 1993-06-29 US disclosed
US-5140023-A Serontonin antagonist; gastrointestinal and psychological disorders; analgesics; antidepressants G. D. SEARLE & CO. (US) 1992-08-18 US disclosed
EP-0454121-A2 Azatetracyclic compounds G.D. Searle & Co. (US) 1991-10-30 EP disclosed