SCHEMBL7307873

SCHEMBL7307873

COC(=O)[C@@H](NC(=O)OCc1cccc(C)n1)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
ALDH1A1 P00352 3/20 0.41
THRB P10828 1/20 0.41
GAA P10253 2/20 0.40
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
TACR3 P29371 1/20 0.39
GRM5 P41594 1/20 0.39
GRM1 Q13255 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
TYR P14679 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298552 0.90 TYR (0.46) MEN1KMT2AOPRM1OPRD1CTSL
SCHEMBL7303071 0.90 TYR (0.46) MEN1KMT2AOPRM1OPRD1CTSL
SCHEMBL4680818 0.81 NPC1 (0.56) ALDH1A1
SCHEMBL3029779 0.81 NPC1 (0.56) ALDH1A1
SCHEMBL7306884 0.80 CYP1A2 (0.48) TACR3
SCHEMBL7306877 0.80 CYP1A2 (0.48) TACR3
SCHEMBL7308154 0.76 CYP3A4 (0.46) CTSBCTSSCTSK
SCHEMBL10535596 0.75 TRPM8 (0.62) MEN1KMT2AALDH1A1CTSLCTSB
SCHEMBL28892051 0.75 TRPM8 (0.62) MEN1KMT2AALDH1A1CTSLCTSB
SCHEMBL10535601 0.75 TRPM8 (0.62) MEN1KMT2AALDH1A1CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed