SCHEMBL7307972

SCHEMBL7307972

COCCN1C(C)=C(C(=O)O)C(c2cccc(C#N)c2Cl)C(C(=O)OC(C)C)=C1C

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PYGM P11217 17/20 0.51
PYGL P06737 16/20 0.51
NR3C2 P08235 2/20 0.42
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752638 1.00 PYGM (0.51) PYGMPYGLNR3C2KDM4E
SCHEMBL5754356 1.00 PYGM (0.51) PYGMPYGLNR3C2KDM4E
SCHEMBL6951169 0.92 NR3C2 (0.43) PYGMPYGLNR3C2KDM4E
SCHEMBL6951538 0.91 PYGM (0.51) PYGMPYGLNR3C2
SCHEMBL9230837 0.90 PYGM (0.51) PYGMPYGLNR3C2
SCHEMBL6947787 0.89 PYGM (0.55) PYGMPYGLNR3C2
SCHEMBL6952771 0.85 NR3C2 (0.42) PYGMPYGLNR3C2
SCHEMBL8877848 0.83 PYGL (0.39) PYGMPYGL
SCHEMBL5080218 0.82 PYGL (0.38) PYGMPYGLNR3C2KDM4E
SCHEMBL5753848 0.81 NR3C2 (0.38) PYGMPYGLNR3C2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657430-B1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1999-06-02 EP claimed
EP-0657430-A1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1995-06-14 EP claimed
EP-0657430-B1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1999-06-02 EP disclosed
EP-0657430-B1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1999-06-02 EP disclosed
EP-0761651-A2 Process for preparing optically active ortho-substituted 4-aryl-dihydropyridines BAYER AG (DE) 1997-03-12 EP disclosed
EP-0657430-A1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1995-06-14 EP disclosed
EP-0657430-A1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1995-06-14 EP disclosed
EP-0657430-A1 Isopropyl-(2-methoxyethyl)-4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-piridine-3,5-dicarboxylate BAYER AG (DE) 1995-06-14 EP disclosed