SCHEMBL7308595

SCHEMBL7308595

CC(C)C[N]C(=O)NCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
KMT2A Q03164 3/20 0.57
MAPT P10636 2/20 0.57
MEN1 O00255 2/20 0.57
L3MBTL1 Q9Y468 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.50
ANPEP P15144 1/20 0.48
HPGD P15428 1/20 0.47
MME P08473 1/20 0.47
GAA P10253 1/20 0.46
SLC1A2 P43004 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL970224 0.81 RIPK1 (0.53) ALDH1A1KMT2AMAPTMEN1L3MBTL1
SCHEMBL969256 0.77 ALDH1A1 (0.55) ALDH1A1KMT2AMAPTMEN1SMN1; SMN2
SCHEMBL4680078 0.77 ALDH1A1 (0.53) ALDH1A1KMT2AMAPTMEN1L3MBTL1
SCHEMBL4680081 0.75 CYP2D6 (0.54) ALDH1A1KMT2AMEN1SMN1; SMN2HPGD
SCHEMBL7351620 0.74 TSHR (0.49) ALDH1A1KMT2AMAPTMEN1
SCHEMBL5866871 0.74 ALDH1A1 (0.71) ALDH1A1KMT2AMAPTMEN1L3MBTL1
SCHEMBL6237639 0.73 ALDH1A1 (0.57) ALDH1A1KMT2AMAPTMEN1L3MBTL1
SCHEMBL27972375 0.73 ALDH1A1 (0.55) ALDH1A1KMT2AMAPTMEN1SMN1; SMN2
SCHEMBL8760 0.73 KMT2A (0.67) ALDH1A1KMT2AMAPTMEN1L3MBTL1
SCHEMBL25379013 0.72 ALDH1A1 (1.00) ALDH1A1KMT2AMAPTMEN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614519-A (1-(2,3 or 4-N-morpholinoalkyl)-imidazol-4-yl)-benizimidazol-1-yl-methyl]-biphenyls useful as angiotensin-II antagonists KARL THOMAE GMBH (DE) 1997-03-25 US disclosed
US-5602127-A ADMINISTERING TO TREAT HYPERTENSION KARL THOMAE GMBH (DE) 1997-02-11 US disclosed
US-5594003-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-14 US disclosed
US-5591762-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5459147-A Angeotensin-antagonistic effects; hypotensive, antiischemic, and antidiabetic agents, treating glaucoma DR. KARL THOMAE GMBH (DE) 1995-10-17 US disclosed
EP-0581166-A1 Benzimidazoles, process for their preparation and their use as angiotensin-II antagonists Dr. Karl Thomae GmbH (DE) 1994-02-02 EP disclosed
EP-0560330-A2 Substituted benzimidazolyl derivatives, therapeutic agents containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-09-15 EP disclosed
EP-0556789-A2 Substituted biphenyl derivatives, therapeutic agents containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-08-25 EP disclosed
EP-0502314-A1 Benzimidazol, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-09 EP disclosed
EP-0470543-A1 Heterocyclic imidazoles, remedies containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-02-12 EP disclosed