SCHEMBL7308747

SCHEMBL7308747

COc1cc(Cl)c([C]=O)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
PDE7A Q13946 1/20 0.34
CYP3A4 P08684 2/20 0.33
MAPT P10636 2/20 0.33
HTR6 P50406 1/20 0.33
LMNA P02545 1/20 0.33
RAF1 P04049 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
GFER P55789 1/20 0.33
PAX8 Q06710 1/20 0.33
RAB9A P51151 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24089350 0.77 ALDH1A1 (0.43) ALDH1A1CYP3A4MAPTLMNAHPGD
SCHEMBL2095222 0.74 ALDH1A1 (0.46) ALDH1A1CYP1A1CYP1B1CYP3A4HPGD
SCHEMBL11595072 0.74 ALDH1A1 (0.46) ALDH1A1CYP1A1CYP1B1CYP3A4HPGD
SCHEMBL7300875 0.73 TAAR1 (0.45) ALDH1A1CYP1A1CYP1B1CYP3A4CA12
SCHEMBL10704960 0.72 ERN1 (0.41) ALDH1A1HSP90AA1CYP3A4MAPTHPGD
SCHEMBL15226652 0.72 ACACB (0.43) HSP90AA1HSP90AB1MAPTRAB9ACA12
SCHEMBL94929 0.72 ALDH1A1 (0.45) ALDH1A1CYP3A4MAPTLMNAHPGD
SCHEMBL1047515 0.72 ALDH1A1 (0.56) ALDH1A1CYP1A1CYP1B1CYP3A4HPGD
SCHEMBL2560197 0.70 ALDH1A1 (0.53) ALDH1A1CYP1A1CYP1B1CYP3A4MAPT
SCHEMBL8430640 0.70 ALDH1A1 (0.53) ALDH1A1CYP1A1CYP1B1CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773456-A EMPHYSEMA, RHEUMATOID ARTHRITIS AND PANCREATITIS SANOFI (FR) 1998-06-30 US disclosed
US-5578623-A DRUGS FOR TREATMENT OF ARTHRITIS, PANCREATITIS, CYSTIC FIBROSIS, BRONCHITIS, RESPIRATORY DISORDERS STERLING WINTHROP INC. (US) 1996-11-26 US disclosed
US-5464852-A Used in treatment of degenerative diseases STERLING WINTHROP INC. (US) 1995-11-07 US disclosed
US-5380737-A Enzyme inhibitors STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0542371-A1 Saccharin derivative proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1993-05-19 EP disclosed