SCHEMBL7309175

SCHEMBL7309175

CC(C)C(C#N)(CCCNC(=O)N1CCC[C@@H]1C(=O)NCc1cccc(Cl)c1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F2 P00734 8/20 0.54
FKBP1A P62942 3/20 0.49
POLB P06746 2/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
CYP2C19 P33261 1/20 0.48
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317230 0.89 F2 (0.63) F2POLBCYP3A4CYP2C9PKM
SCHEMBL7317235 0.89 F2 (0.63) F2POLBCYP3A4CYP2C9PKM
SCHEMBL7316567 0.84 FKBP1A (0.48) FKBP1APOLBCYP3A4CYP2C9PKM
SCHEMBL7306123 0.82 CFD (0.47) FKBP1ACYP3A4CYP2C9PKMCYP2C19
SCHEMBL7316804 0.81 F2 (0.51) F2FKBP1APOLBCYP3A4CYP2C9
SCHEMBL7316811 0.81 F2 (0.51) F2FKBP1APOLBCYP3A4CYP2C9
SCHEMBL7305369 0.81 F2 (0.51) F2FKBP1APOLBCYP3A4CYP2C9
SCHEMBL7305382 0.81 F2 (0.51) F2FKBP1APOLBCYP3A4CYP2C9
SCHEMBL7306032 0.81 F2 (0.49) F2FKBP1APOLBCYP3A4CYP2C9
SCHEMBL7306042 0.81 F2 (0.49) F2FKBP1APOLBCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed