SCHEMBL7309575

SCHEMBL7309575

CC(CCCNC(CC1CCCCC1)C(=O)CSCc1ccco1)N(C)C(=O)COc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
HPGD P15428 3/20 0.41
MAPT P10636 2/20 0.41
POLB P06746 2/20 0.41
USP2 O75604 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPY5R Q15761 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GPR88 Q9GZN0 1/20 0.37
TSHR P16473 1/20 0.34
REN P00797 3/20 0.33
MMP3 P08254 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311207 0.87 ALDH1A1 (0.45) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7301637 0.86 ALDH1A1 (0.44) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7303790 0.86 ALDH1A1 (0.44) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7302476 0.86 MAPT (0.44) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7315651 0.84 MAPT (0.46) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7444212 0.83 ALDH1A1 (0.42) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7309565 0.78 REN (0.46) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7309584 0.78 REN (0.46) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7309585 0.76 ALDH1A1 (0.47) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7303759 0.76 ALDH1A1 (0.40) ALDH1A1HPGDMAPTPOLBUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed