SCHEMBL7309612

SCHEMBL7309612

CCn1nc(-c2cccc(Br)c2)cc(Nc2ccnc3ccccc23)c1=O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.52
EGFR P00533 2/20 0.50
RIPK2 O43353 1/20 0.41
ALK Q9UM73 2/20 0.40
LMNA P02545 2/20 0.40
MKNK1 Q9BUB5 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
MITF O75030 1/20 0.39
RAD52 P43351 1/20 0.39
HTR2C P28335 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306528 0.94 PDE4B (0.52) PDE4BEGFRLMNAALDH1A1ADORA2A
SCHEMBL4052027 0.86 PDE4B (0.54) PDE4BLMNAALDH1A1HTR2CMEN1
SCHEMBL4049841 0.82 TBXAS1 (0.49) PDE4BRIPK2LMNAADORA2AADORA2B
SCHEMBL4056450 0.81 PDE4B (0.46) PDE4BLMNAALDH1A1ADORA2AADORA2B
SCHEMBL7316209 0.80 PDE4B (0.61) PDE4BADORA2AADORA2BADORA1
SCHEMBL4050499 0.80 PDE4B (0.46) PDE4BLMNAALDH1A1HTR2CMEN1
SCHEMBL7314230 0.79 PDE4B (0.52) PDE4BADORA2AADORA2BADORA1
SCHEMBL7308904 0.79 PDE4B (0.56) PDE4BADORA2AADORA2BADORA1MEN1
SCHEMBL4055355 0.78 RECQL (0.51) PDE4BHTT
SCHEMBL7304940 0.78 PDE4B (0.59) PDE4BADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394998-A1 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3-yl)-biphenyl derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-12-14 EP disclosed