SCHEMBL7310776

SCHEMBL7310776

CC(C)C(C#N)(CCCCC(=O)N1CCC[C@@H]1C(=O)NCCc1ccc([N+](=O)[O-])cc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 2/20 0.41
PKM P14618 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
POLB P06746 1/20 0.41
F2 P00734 2/20 0.41
FKBP1A P62942 3/20 0.41
ITGB1 P05556 4/20 0.40
ITGA4 P13612 4/20 0.40
ATM Q13315 1/20 0.40
MEN1 O00255 1/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CHRM3 P20309 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310783 1.00 CYP3A4 (0.42) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL7318694 0.93 DPP4 (0.44) CYP3A4CYP2C9PKMPOLBF2
SCHEMBL7318701 0.93 DPP4 (0.44) CYP3A4CYP2C9PKMPOLBF2
SCHEMBL7301363 0.92 FKBP1A (0.47) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL7301358 0.92 FKBP1A (0.47) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL7305475 0.88 FKBP1A (0.53) F2FKBP1AITGB1ITGA4DPP4
SCHEMBL7305485 0.88 FKBP1A (0.53) F2FKBP1AITGB1ITGA4DPP4
SCHEMBL7309531 0.87 FKBP1A (0.51) F2FKBP1AITGB1ITGA4
SCHEMBL7309517 0.87 FKBP1A (0.51) F2FKBP1AITGB1ITGA4
SCHEMBL7316065 0.85 DPP4 (0.48) KMT2APOLBF2FKBP1AITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed