SCHEMBL7310951

SCHEMBL7310951

CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)COc1c(Cl)cc(Cl)cc1Cl)C(=O)CSCc1ccco1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
HPGD P15428 5/20 0.44
MAPT P10636 5/20 0.44
POLB P06746 4/20 0.44
USP2 O75604 3/20 0.44
HSD17B10 Q99714 2/20 0.44
LMNA P02545 2/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
ALOX12 P18054 1/20 0.44
ATM Q13315 1/20 0.44
CASP3 P42574 4/20 0.41
CASP1 P29466 3/20 0.41
CASP7 P55210 3/20 0.41
CASP6 P55212 3/20 0.41
CASP8 Q14790 3/20 0.41
RAB9A P51151 3/20 0.40
TDP1 Q9NUW8 3/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310961 1.00 ALDH1A1 (0.44) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7301044 0.92 HPGD (0.49) ALDH1A1HPGDMAPTPOLBLMNA
SCHEMBL7301037 0.92 HPGD (0.49) ALDH1A1HPGDMAPTPOLBLMNA
SCHEMBL7304720 0.90 ALDH1A1 (0.40) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7436035 0.90 ALDH1A1 (0.40) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7441563 0.89 POLB (0.40) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7441573 0.89 POLB (0.40) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7310960 0.89 ALDH1A1 (0.42) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7312214 0.88 ALDH1A1 (0.38) ALDH1A1HPGDMAPTPOLBUSP2
SCHEMBL7312203 0.88 ALDH1A1 (0.38) ALDH1A1HPGDMAPTPOLBUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed