SCHEMBL7310985

SCHEMBL7310985

CCCc1nc(CO)c(C(=O)OCC)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 11/20 0.61
AGTR2 P50052 10/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1417588 0.92 AGTR1 (0.67) AGTR1AGTR2
SCHEMBL3841141 0.90 AGTR1 (0.65) AGTR1AGTR2
SCHEMBL669229 0.90 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL9389798 0.89 AGTR1 (0.64) AGTR1AGTR2
SCHEMBL9198706 0.89 AGTR1 (0.62) AGTR1AGTR2
SCHEMBL986792 0.88 AGTR1 (0.62) AGTR1AGTR2
SCHEMBL7302931 0.88 AGTR1 (0.56) AGTR1AGTR2
SCHEMBL7304486 0.88 AGTR1 (0.57) AGTR1AGTR2
SCHEMBL669266 0.88 AGTR2 (0.66) AGTR1AGTR2
Hydrochloric Acid SCHEMBL7305266 0.88 AGTR1 (0.62) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545912-B1 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0545912-A2 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1993-06-09 EP disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed