SCHEMBL7311003

SCHEMBL7311003

COCOc1cc(COC(=O)O)on1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.38
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMPD1 P17405 1/20 0.36
SLC6A2 P23975 1/20 0.36
HTR2A P28223 1/20 0.36
SLC6A3 Q01959 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303479 0.77 NOTUM (0.43)
SCHEMBL13762097 0.75 MEN1 (0.37) NPC1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL7311748 0.72 SMPD1 (0.46) MRGPRX4NPC1RAB9ASMPD1MAPT
SCHEMBL13754957 0.72 SMPD1 (0.43) NPC1RAB9AL3MBTL1SMPD1MAPT
SCHEMBL189694 0.70 SMN1; SMN2 (0.53) NPC1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL1416805 0.70 ALDH1A1 (0.48) NPC1POLBRAB9AMAPT
SCHEMBL8378803 0.69 CHRM4 (0.50) NPC1POLBRAB9ASMN1; SMN2L3MBTL1
SCHEMBL9134303 0.67 HCAR2 (0.50) MRGPRX4NPC1POLBRAB9ASMN1; SMN2
SCHEMBL10415792 0.67 KDM4E (0.46) RAB9A
SCHEMBL8121102 0.67 HRH3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed