SCHEMBL7311364

SCHEMBL7311364

c1nc2cnc(N3CCNCC3)nc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.47
CASP1 P29466 14/20 0.47
CYP1A2 P05177 13/20 0.47
CASP7 P55210 13/20 0.47
HSD17B10 Q99714 13/20 0.47
HPGD P15428 8/20 0.47
CYP3A4 P08684 6/20 0.47
TSHR P16473 3/20 0.47
CYP2C19 P33261 3/20 0.47
KDM4E B2RXH2 1/20 0.43
USP2 O75604 5/20 0.43
CYP2C9 P11712 6/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HRH1 P35367 1/20 0.42
GLA P06280 3/20 0.41
HIF1A Q16665 3/20 0.41
TAAR1 Q96RJ0 1/20 0.41
ADRB1 P08588 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11611665 0.87 IP6K1 (0.44) ALDH1A1CASP1TSHRUSP2HRH1
SCHEMBL15322620 0.85 IP6K1 (0.43) ALDH1A1TSHRUSP2ALOX15SMN1; SMN2
SCHEMBL336705 0.83 KDM4E (0.49) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL30677292 0.83 KDM4E (0.49) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL30945083 0.74 ROCK2 (0.50) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL2508000 0.74 SCD (0.49) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL7269241 0.73 ROCK2 (0.50) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL6070116 0.73 PDE4A (0.46) ALDH1A1CASP1KDM4EUSP2KMT2A
Hydrochloric Acid SCHEMBL6017462 0.73 ROCK2 (0.49) ALDH1A1CASP1CYP1A2CASP7HSD17B10
SCHEMBL291823 0.72 ALDH1A1 (0.49) ALDH1A1CASP1CYP1A2CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0331511-B1 6-SUBSTITUTED PURINYL PIPERAZINE DERIVATIVES ORTHO PHARMACEUTICAL CORPORATION (US) 1993-07-28 EP disclosed
EP-0458618-A1 6-Substituted purinyl piperazine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1991-11-27 EP disclosed
EP-0331511-A1 6-Substituted purinyl piperazine derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1989-09-06 EP disclosed