SCHEMBL7312700

SCHEMBL7312700

CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)Cc1cccc2ccccc12)C(=O)CSCc1ccco1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.47
CASP3 P42574 2/20 0.47
CASP7 P55210 2/20 0.47
ANPEP P15144 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
REN P00797 3/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
MCHR1 Q99705 1/20 0.39
MME P08473 1/20 0.38
ACE P12821 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
PSMB5 P28074 3/20 0.38
LCK P06239 2/20 0.38
CASP6 P55212 1/20 0.38
CASP8 Q14790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307336 0.88 PSMB5 (0.47) CASP1CASP3CASP7ANPEPALDH1A1
SCHEMBL7305782 0.87 MCHR1 (0.41) CASP1CASP3CASP7ALDH1A1MCHR1
SCHEMBL7305792 0.87 MCHR1 (0.41) CASP1CASP3CASP7ALDH1A1MCHR1
SCHEMBL7312916 0.87 POLB (0.46) CASP1CASP3ALDH1A1PSMB5POLB
SCHEMBL7312904 0.87 POLB (0.46) CASP1CASP3ALDH1A1PSMB5POLB
SCHEMBL7302087 0.85 POLB (0.40) CASP1CASP3CASP7ALDH1A1PSMB5
SCHEMBL7305772 0.85 PSMB5 (0.37) ALDH1A1PSMB5POLBHPGDMMP9
SCHEMBL7434956 0.83 MMP3 (0.36) CASP1CASP3CASP7ANPEPALDH1A1
SCHEMBL7302479 0.83 ALDH1A1 (0.48) CASP1CASP3CASP7ALDH1A1REN
SCHEMBL7311282 0.83 ALDH1A1 (0.43) CASP1CASP3ANPEPALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed