SCHEMBL7313985

SCHEMBL7313985

CCOC(=O)CC(C(=O)OCC)N1CCN(CC2CN(c3ccc(C(=N)N)cc3)C(=O)O2)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.60
ITGA2B P08514 11/20 0.60
PRSS1 P07477 9/20 0.51
PRSS2 P07478 9/20 0.51
PRSS3 P35030 9/20 0.51
F10 P00742 8/20 0.50
F2 P00734 1/20 0.43
SIGMAR1 Q99720 6/20 0.41
GRM2 Q14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858188 0.94 ITGB3 (0.55) ITGB3ITGA2BPRSS1PRSS2PRSS3
Acetic Acid SCHEMBL8858146 0.93 ITGB3 (0.54) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7305905 0.90 ITGB3 (0.65) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7305481 0.89 ITGB3 (0.55) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7316851 0.88 ITGB3 (0.54) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948638 0.87 ITGB3 (0.75) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948633 0.87 ITGB3 (0.75) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8948635 0.87 ITGB3 (0.75) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7306506 0.86 ITGB3 (0.52) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7316531 0.85 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5627197-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-05-06 US claimed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP claimed
US-5627197-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-05-06 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed