SCHEMBL7314949

SCHEMBL7314949

CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)NCc1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
P2RX7 Q99572 1/20 0.56
HRH3 Q9Y5N1 1/20 0.55
KMT2A Q03164 3/20 0.53
TSHR P16473 1/20 0.53
KDM4E B2RXH2 1/20 0.52
TACR1 P25103 2/20 0.51
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
F2 P00734 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPC1 O15118 1/20 0.49
MEN1 O00255 2/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
CYP2C19 P33261 1/20 0.48
USP30 Q70CQ3 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989544 0.91 ALDH1A1 (0.66) ALDH1A1KMT2AKDM4ELMNANPSR1
SCHEMBL893264 0.90 ALDH1A1 (0.54) ALDH1A1P2RX7HRH3KMT2ATSHR
SCHEMBL29514072 0.90 ALDH1A1 (0.54) ALDH1A1P2RX7HRH3KMT2ATSHR
SCHEMBL17056182 0.90 ALDH1A1 (0.54) ALDH1A1P2RX7HRH3KMT2ATSHR
SCHEMBL18882738 0.87 ALDH1A1 (0.51) ALDH1A1P2RX7HRH3KMT2ATSHR
SCHEMBL15681742 0.87 WNT3 (0.54) ALDH1A1HRH3KMT2ALMNANPSR1
SCHEMBL17056184 0.86 ALDH1A1 (0.56) ALDH1A1KMT2ATACR1LMNANPSR1
SCHEMBL29513950 0.86 ALDH1A1 (0.61) ALDH1A1KMT2AKDM4ELMNANPSR1
SCHEMBL7307776 0.86 ALDH1A1 (0.72) ALDH1A1P2RX7KMT2ALMNANPSR1
SCHEMBL17056181 0.86 ALDH1A1 (0.61) ALDH1A1KMT2AKDM4ELMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed