SCHEMBL7315722

SCHEMBL7315722

C=CCOCc1cccc(OCC(O)CNC(C)(C)Cc2ccccc2)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.59
CYP2D6 P10635 3/20 0.48
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
ADRB2 P07550 1/20 0.45
ADRB3 P13945 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316623 0.90 CASR (0.66) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7310724 0.89 CYP2D6 (0.56) CASRCYP2D6ADRB2ADRB3
SCHEMBL7306704 0.83 CYP2D6 (0.62) CYP2D6SLC6A2SLC6A4KCNH2ADRB2
SCHEMBL7317233 0.83 CASR (0.59) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7312172 0.82 ADRB3 (0.55) ADRB2ADRB3
SCHEMBL14383031 0.81 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL5510479 0.80 CASR (0.81) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL14383077 0.79 CASR (0.78) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7318229 0.78 CASR (0.56) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL11513676 0.78 CYP2D6 (0.50) CYP2D6SLC6A4ADRB2ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed