SCHEMBL7318229

SCHEMBL7318229

C=CCOCCOCc1ccccc1OCC(O)CNC(C)(C)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 9/20 0.56
ADRB2 P07550 10/20 0.47
ADRB1 P08588 4/20 0.47
HTR1A P08908 4/20 0.47
CYP2D6 P10635 4/20 0.47
ADRB3 P13945 4/20 0.47
SLC6A4 P31645 3/20 0.47
LMNA P02545 3/20 0.47
SLC6A2 P23975 2/20 0.47
KCNH2 Q12809 2/20 0.47
ADRA1A P35348 2/20 0.47
CYP1A2 P05177 2/20 0.47
ADRA2C P18825 1/20 0.47
BDKRB2 P30411 1/20 0.47
HTR2B P41595 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KDM4E B2RXH2 1/20 0.47
PMP22 Q01453 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317233 0.95 CASR (0.59) CASRADRB2ADRB1HTR1ACYP2D6
SCHEMBL7319524 0.88 CASR (0.60) CASRADRB2ADRB1CYP2D6ADRB3
SCHEMBL7308129 0.88 MAPT (0.53) ADRB2ADRB1HTR1ACYP2D6ADRB3
SCHEMBL7318237 0.86 CASR (0.56) CASRADRB2HTR1ACYP2D6ADRB3
SCHEMBL7319712 0.86 CASR (0.58) CASRADRB2ADRB1CYP2D6ADRB3
SCHEMBL7319028 0.83 ADRB2 (0.56) ADRB2ADRB1HTR1ACYP2D6ADRB3
SCHEMBL7312061 0.83 ADRB2 (0.69) ADRB2ADRB1HTR1ACYP2D6ADRB3
SCHEMBL7310963 0.82 MAPT (0.56) ADRB2ADRB1HTR1ACYP2D6ADRB3
SCHEMBL11511416 0.81 CASR (0.59) CASRADRB2CYP2D6ADRB3SLC6A4
SCHEMBL11522955 0.80 ADRB2 (0.62) CASRADRB2ADRB1HTR1ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed