SCHEMBL7315776

SCHEMBL7315776

COc1ccc(CCc2cc(F)cc(CCCN(C)OC(=O)C(=O)O)c2I)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTR2A P28223 5/20 0.41
HTR2C P28335 5/20 0.41
HTR2B P41595 5/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
SMPD1 P17405 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
AOC3 Q16853 1/20 0.39
ABCB1 P08183 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL10690881 0.73 ALDH1A1 (0.55) KDM4EALDH1A1HTR2AHTR2CHTR2B
SCHEMBL31123655 0.65 ATM (0.49) KDM4EABCB1KMT2AMEN1
SCHEMBL7356879 0.65 CDK8 (0.61) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL9781645 0.65 CYP1A2 (0.56) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL3345442 0.64 CYP1A2 (0.64) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL10426074 0.64 KMT2A (0.60) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
Oxalic Acid SCHEMBL7274490 0.63 CYP3A4 (0.67) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL27572903 0.63 CHRM5 (0.52) KDM4EALDH1A1HTR2AHTR2CHTR2B
SCHEMBL31157848 0.63 CYP19A1 (0.77) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL16641094 0.63 CYP19A1 (0.77) KDM4EALDH1A1CYP3A4CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed