SCHEMBL7315795

SCHEMBL7315795

COc1ccc(I)c(CC(C)NCCc2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
SLC2A1 P11166 2/20 0.47
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SIGMAR1 Q99720 3/20 0.46
HTR2A P28223 3/20 0.41
SLC6A4 P31645 3/20 0.41
KCNH2 Q12809 2/20 0.41
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
CASR P41180 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317493 0.85 SLC2A1 (0.52) MEN1KMT2ASLC2A1HTTSMN1; SMN2
SCHEMBL9825369 0.85 KCNH2 (0.50) MEN1KMT2ASLC2A1HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL7320769 0.84 KCNH2 (0.49) MEN1KMT2ASLC2A1HTTSMN1; SMN2
SCHEMBL9825118 0.83 SLC2A1 (0.43) MEN1KMT2ASLC2A1HTTSMN1; SMN2
SCHEMBL9824522 0.79 SLC2A1 (0.48) MEN1KMT2ASLC2A1HTTSMN1; SMN2
SCHEMBL9824218 0.79 SLC2A1 (0.48) MEN1KMT2ASLC2A1HTTSMN1; SMN2
SCHEMBL7312568 0.79 SIGMAR1 (0.47) MEN1KMT2ASLC2A1HTTSMN1; SMN2
Fumaric Acid SCHEMBL7311253 0.78 ALDH1A1 (0.42) MEN1KMT2ASLC2A1HTTSMN1; SMN2
Fumaric Acid SCHEMBL10690449 0.75 SLC2A1 (0.40) MEN1KMT2ASLC2A1SIGMAR1HTR2A
SCHEMBL14438281 0.70 SIGMAR1 (0.54) MEN1KMT2ASIGMAR1KCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed