SCHEMBL7316115

SCHEMBL7316115

COc1ccc(C2(O[C@H](C)[C@H](N)C(=O)O)c3ccccc3-c3ccccc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.45
SLC6A12 P48065 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316108 1.00 KIF11 (0.45) KIF11SLC6A12NPC1MAPTMAPK1
SCHEMBL7325057 0.91 PDK2 (0.43) KIF11SLC6A12KMT2APDK2
SCHEMBL7325065 0.91 PDK2 (0.43) KIF11SLC6A12KMT2APDK2
SCHEMBL7317367 0.90 KIF11 (0.44) KIF11MAPTKMT2ASLC1A3SLC1A2
SCHEMBL7317362 0.90 KIF11 (0.44) KIF11MAPTKMT2ASLC1A3SLC1A2
SCHEMBL7323867 0.90 KIF11 (0.44) KIF11MAPTKMT2ASLC1A3SLC1A2
SCHEMBL7323752 0.87 KIF11 (0.37) KIF11MAPTPDK2
SCHEMBL7323759 0.87 KIF11 (0.37) KIF11MAPTPDK2
SCHEMBL7318078 0.86 CYP2C19 (0.49) KIF11KMT2APDK2
SCHEMBL7323278 0.86 KIF11 (0.49) KIF11NPC1KMT2ASLC1A3SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO claimed
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed