SCHEMBL7316116

SCHEMBL7316116

COc1cccc(OC)c1C[N@+]1(C(=O)CCCC[C@@](C#N)(c2ccccc2)C(C)C)CCCC1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.38
ABCB1 P08183 10/20 0.35
CYP3A4 P08684 7/20 0.35
EBP Q15125 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
TSHR P16473 3/20 0.33
LMNA P02545 3/20 0.33
KCNH2 Q12809 3/20 0.33
HTR1A P08908 3/20 0.33
MAPK1 P28482 2/20 0.33
CACNA1F O60840 2/20 0.33
ADRA2A P08913 2/20 0.33
DRD2 P14416 2/20 0.33
ADRA2C P18825 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
SLC6A4 P31645 2/20 0.33
DRD3 P35462 2/20 0.33
SCN1A P35498 2/20 0.33
HTR2B P41595 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317309 0.92 CACNA1B (0.37) CACNA1BABCB1CYP3A4EBPSIGMAR1
SCHEMBL7314456 0.89 ABCB1 (0.42) CACNA1BABCB1CYP3A4EBPSIGMAR1
SCHEMBL7315667 0.88 CACNA1B (0.38) CACNA1BABCB1CYP3A4EBPSIGMAR1
SCHEMBL7306036 0.88 EBP (0.41) CACNA1BEBPSIGMAR1
SCHEMBL7301603 0.88 CACNA1B (0.36) CACNA1BABCB1CYP3A4EBPSIGMAR1
SCHEMBL7313731 0.87 CACNA1B (0.38) CACNA1BABCB1CYP3A4EBPSIGMAR1
SCHEMBL7309087 0.86 CACNA1B (0.34) CACNA1BABCB1EBPSIGMAR1
SCHEMBL7311990 0.86 EBP (0.33) CACNA1BEBPSIGMAR1DRD2DRD3
SCHEMBL7309476 0.86 EBP (0.36) CACNA1BEBPSIGMAR1
SCHEMBL7302555 0.85 EBP (0.33) CACNA1BEBPSIGMAR1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed