SCHEMBL7316245

SCHEMBL7316245

COC(=O)c1ccc(Cl)c(C)c1N(Cc1ccccc1)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 16/20 0.64
MMP1 P03956 15/20 0.64
MMP13 P45452 16/20 0.60
ADAM17 P78536 5/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
NR3C1 P04150 1/20 0.52
PGR P06401 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7312470 0.92 MMP9 (0.63) MMP9MMP1MMP13ADAM17ALDH1A1
SCHEMBL7317324 0.90 MMP9 (0.79) MMP9MMP1MMP13ADAM17
SCHEMBL7319113 0.88 MMP9 (0.81) MMP9MMP1MMP13ADAM17NR3C1
SCHEMBL7321969 0.82 MMP9 (0.66) MMP9MMP1MMP13ADAM17ALDH1A1
SCHEMBL7504875 0.82 MMP9 (0.68) MMP9MMP1MMP13ADAM17
SCHEMBL7317407 0.82 MMP13 (0.83) MMP9MMP1MMP13ADAM17ALDH1A1
SCHEMBL28741388 0.81 MMP13 (0.58) MMP9MMP1MMP13ADAM17ALDH1A1
SCHEMBL7313797 0.81 MMP13 (0.72) MMP9MMP1MMP13ADAM17
SCHEMBL7316528 0.80 MMP13 (0.69) MMP9MMP1MMP13ADAM17NR3C1
SCHEMBL7446307 0.80 MMP13 (0.68) MMP9MMP1MMP13ADAM17ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP disclosed
CN-1240429-A Preparation and use of ortho-sulfonamido aryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors AMERICAN CYANAMID CO (US) 2000-01-05 CN disclosed
EP-0938471-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-09-01 EP disclosed
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed
WO-1998016503-A2 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO disclosed