SCHEMBL7316490

SCHEMBL7316490

N=C(N)c1nc(-c2cccc(C(F)(F)F)c2)cs1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
CFTR P13569 2/20 0.52
AR P10275 1/20 0.50
ADAM17 P78536 1/20 0.50
ITGB3 P05106 4/20 0.48
ITGA2B P08514 4/20 0.48
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
SCN9A Q15858 1/20 0.46
C1S P09871 1/20 0.46
LTA4H P09960 1/20 0.46
IDO1 P14902 1/20 0.46
CASP3 P42574 1/20 0.46
CASP7 P55210 1/20 0.46
CASP8 Q14790 1/20 0.46
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440522 0.86 CYP3A4 (0.61) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL7426086 0.84 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL7426082 0.84 MEN1 (0.51) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL3749301 0.82 ALDH1A1 (0.67) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL13078605 0.81 ALDH1A1 (0.59) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL3609002 0.81 CFTR (0.60) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL474410 0.80 LTA4H (0.67) ALDH1A1KDM4EMEN1KMT2ACFTR
Bromide SCHEMBL8357468 0.79 LTA4H (0.65) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL13044095 0.78 ALDH1A1 (0.56) ALDH1A1KDM4EMEN1KMT2ACFTR
SCHEMBL1198896 0.77 ALDH1A1 (0.56) ALDH1A1KDM4EMEN1KMT2ACFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665724-A Substituted pyrimidinylaminothiazole derivatives useful as platelet aggregation inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1997-09-09 US disclosed
US-5530000-A Substituted pyrimidinylaminothiazole derivatives useful as platelet aggreggation inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1996-06-25 US disclosed
US-5405848-A Substituted thiazolylaminotetrahydropyridopyrimidines derivatives useful as platelet aggregation inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1995-04-11 US disclosed