SCHEMBL7316679

SCHEMBL7316679

Cc1cc(C)c(N(Cc2ccccc2)S(=O)(=O)c2ccc(OCc3ccccc3)cc2)c(C(=O)NO)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 19/20 1.00
MMP9 P14780 16/20 1.00
ADAM17 P78536 10/20 1.00
MMP1 P03956 14/20 0.85
TDP1 Q9NUW8 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310743 0.93 MMP13 (0.94) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL7317442 0.92 MMP13 (1.00) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL7325555 0.91 MMP13 (0.83) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL6129978 0.90 MMP13 (1.00) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL7319243 0.90 MMP13 (0.93) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL7453410 0.90 MMP13 (1.00) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL6129964 0.90 MMP13 (1.00) MMP13MMP9ADAM17MMP1
SCHEMBL6129934 0.90 MMP13 (0.84) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL6129932 0.90 MMP13 (0.81) MMP13MMP9ADAM17MMP1TDP1
SCHEMBL3949565 0.88 MMP13 (0.78) MMP13MMP9ADAM17MMP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP claimed
EP-0938471-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-09-01 EP claimed
WO-1998016503-A2 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO claimed
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP disclosed
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed