SCHEMBL7318927

SCHEMBL7318927

COc1ccc(CC(Cl)NCc2ccccc2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.55
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
KMT2A Q03164 3/20 0.51
LDHA P00338 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.48
ATM Q13315 1/20 0.48
MEN1 O00255 2/20 0.48
PPARA Q07869 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PPARG P37231 1/20 0.46
KDM1A O60341 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929023 0.84 SIGMAR1 (0.63) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL7929020 0.84 SIGMAR1 (0.63) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL5022424 0.81 SMN1; SMN2 (0.52) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL10961223 0.79 SIGMAR1 (0.51) LDHAATMSIGMAR1
SCHEMBL6095764 0.78 KMT2A (0.63) SMN1; SMN2LMNAMAPTKMT2AALDH1A1
SCHEMBL6095767 0.78 KMT2A (0.63) SMN1; SMN2LMNAMAPTKMT2AALDH1A1
SCHEMBL4888632 0.78 LDHA (0.55) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL4888641 0.78 LDHA (0.55) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL4891278 0.78 LDHA (0.55) SMN1; SMN2LMNAMAPTKMT2ALDHA
SCHEMBL29207901 0.77 SMN1; SMN2 (0.66) SMN1; SMN2LMNAMAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359464-A 3-Furylmethyl-6-halo-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines and antihypertensive use thereof SMITHKLINE BECKMAN CORPORATION (US) 1982-11-16 US disclosed
US-4352754-A HYPOTENSIVE, ANTI-PARKINSON SMITHKLINE CORPORATION (US) 1982-10-05 US disclosed
US-4255422-A DIURETICS, TREATMENT OF CARDIOVASCULAR DISORDERS SMITHKLINE CORPORATION (US) 1981-03-10 US disclosed
US-4192872-A ANTI -PARKINSONISM ACTIVITY SMITHKLINE CORPORATION (US) 1980-03-11 US disclosed
US-4160765-A Method for 6-bromination of 1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine compounds SMITHKLINE CORPORATION (US) 1979-07-10 US disclosed