SCHEMBL7319618

SCHEMBL7319618

CCOC(=O)CNC(=O)C(Cc1ccc(-c2ccccc2)cc1)N(CP(=O)(O)O)C(OC(=O)CC)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPID Q08752 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ABCC3 O15438 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
NR3C1 P04150 1/20 0.37
RARG P13631 1/20 0.37
CNR1 P21554 1/20 0.37
OPRK1 P41145 1/20 0.37
NR1H2 P55055 1/20 0.37
PPARA Q07869 1/20 0.37
NR1H3 Q13133 1/20 0.37
NR1I3 Q14994 1/20 0.37
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MME P08473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311798 0.81 HDAC3 (0.37)
SCHEMBL7317919 0.81 PPID (0.41) PPIDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7311117 0.79 MMEL1 (0.37) EED
SCHEMBL7321202 0.79 MME (0.40) MMEANPEP
SCHEMBL7349076 0.78 MMEL1 (0.44)
SCHEMBL7320395 0.78 MMEL1 (0.44)
SCHEMBL7316906 0.78 CYP3A4 (0.40) CYP3A4CYP2D6CYP2C19
SCHEMBL7318600 0.76 MMEL1 (0.39) CYP3A4CYP2D6CYP2C19MAPTRAB9A
SCHEMBL7319612 0.74 MME (0.38) PPIDMAPTRAB9AMMEKLKB1
SCHEMBL7312623 0.74 MMEL1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP claimed
EP-0592367-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1994-04-13 EP disclosed
US-5294632-A Diuretics and vasorelaxants CIBA-GEIGY CORPORATION (US) 1994-03-15 US disclosed
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP disclosed
US-5155100-A Treating cardiovascular disorders in mammals CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed