SCHEMBL7319792

SCHEMBL7319792

C=CCOCc1ccc(OCC(O)CNC(C)CO)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.60
ADRB3 P13945 8/20 0.56
ADRB2 P07550 8/20 0.56
ADRB1 P08588 6/20 0.56
MEN1 O00255 2/20 0.49
LMNA P02545 2/20 0.49
KMT2A Q03164 2/20 0.49
THRB P10828 1/20 0.49
ALOX12 P18054 1/20 0.49
NFKB1 P19838 1/20 0.49
APEX1 P27695 1/20 0.49
MAPK1 P28482 1/20 0.49
PTGS1 P23219 1/20 0.49
SLC6A2 P23975 1/20 0.49
ADRA1A P35348 2/20 0.46
SLC22A1 O15245 1/20 0.46
CYP1A2 P05177 1/20 0.46
HTR1A P08908 1/20 0.46
HTR2A P28223 1/20 0.46
SLC6A4 P31645 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307918 0.89 CYP2D6 (0.76) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL11513676 0.87 CYP2D6 (0.50) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL7306755 0.81 ADRB3 (0.80) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL7315332 0.81 ADRB2 (0.60) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL11512576 0.80 ADRB2 (0.60) CYP2D6ADRB3ADRB2ADRB1LMNA
SCHEMBL5351511 0.78 CYP2D6 (0.73) CYP2D6ADRB2ADRB1MEN1LMNA
SCHEMBL5852432 0.78 CYP2D6 (0.73) CYP2D6ADRB2ADRB1MEN1LMNA
SCHEMBL7313076 0.77 CYP2D6 (0.47) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL7318192 0.77 CYP2D6 (0.47) CYP2D6ADRB3ADRB2ADRB1MEN1
SCHEMBL28403894 0.77 ADRB2 (0.78) CYP2D6ADRB3ADRB2ADRB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed